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Ketoconazole

Ketoconazole

Ketoconazole, igurishwa ku izina rya Nizoral n'indi, ni umuti uvura indwara ziterwa n'imiti irwanya udukoko ukoreshwa mu kuvura indwara zitandukanye z'imiti. Iyo ikoreshejwe ku ruhu, ikoreshwa mu kuvura indwara z'uruhu ziterwa n'ibihumyo nka tinea, candidiasis y'uruhu, pityriasis versicolor, dandruff, na seborrheic dermatitis. Iyo uyinyoye ntabwo ari amahitamo meza cyane kandi ni byiza kuyikoresha gusa ku ndwara zikomeye mu gihe izindi miti zidashobora gukoreshwa. Izindi ngamba zirimo kuvura imikurire y'umusatsi ikabije ndetse n'indwara ya Cushing's syndrome.

Ingaruka mbi zikunze kugaragara iyo zikoreshejwe ku ruhu zirimo gutukura, kuribwa no kuruma. Ingaruka mbi zikunze kugaragara iyo umuntu anyoye zirimo isesemi, kuribwa umutwe, n'ibibazo by'umwijima. Ibibazo by'umwijima bishobora gutera urupfu cyangwa gukenera guterwa umwijima. Izindi ngaruka mbi zikomeye iyo umuntu anyoye zirimo gukomeretsa QT, kudakora neza kw'uturemangingo tw'amaraso, no kunanirwa k'umubiri. Ni imidazole kandi ikora mu kugira ingaruka ku ikorwa rya ergosterol ikenewe ku ruhu rw'uturemangingo tw'ibihumyo bityo igatuma gukura kugabanuka.

Ketoconazole yahawe uburenganzira bwo gukoresha imiti mu 1977, itangira gukoreshwa mu buvuzi mu 1981. Iraboneka nk'umuti usanzwe kandi imiti ikoreshwa ku ruhu igurishwa ku giciro cya muganga mu Bwongereza. Umuyoboro wa garama 30 mu Bwongereza utwara NHS munsi y'amapawundi 5 mu 2019. Muri Leta Zunze Ubumwe za Amerika, aho amavuta yo mu bwoko bwa "topical cream" aboneka gusa ku muganga, ikiguzi cy'aya mafaranga ni hafi US$6.30. Mu 2017, wari umuti wa 219 ukunze kwandikirwa muri Leta Zunze Ubumwe za Amerika, aho wanditswe n'abaganga barenga miliyoni ebyiri. Iyi ngingo ifatwa mu kanwa yakuweho mu Muryango w’Ubumwe bw’u Burayi no muri Ositaraliya mu 2013 no mu Bushinwa mu 2015. Byongeye kandi, ikoreshwa ryayo ryaragabanijwe muri Leta Zunze Ubumwe za Amerika na Kanada mu 2013.

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Text from Wikipedia, CC BY-SA 4.0 · Source article